SCHEMBL5239771

SCHEMBL5239771

Cc1nc2ccc(N3CCC(O)(c4ccccc4)CC3)cc2c(-c2ccc(F)cc2)c1C(F)(F)C(=O)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.42
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.37
MC4R P32245 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
DRD2 P14416 1/20 0.35
CASP3 P42574 1/20 0.34
FABP3 P05413 1/20 0.34
FABP4 P15090 1/20 0.34
PRNP P04156 1/20 0.34
PPARG P37231 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NR2E3 Q9Y5X4 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
AR P10275 1/20 0.34
KCNH2 Q12809 1/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27685125 0.87 MCHR1 (0.38) MCHR1ALDH1A1TP53MC4ROPRM1
SCHEMBL2828012 0.85 ALDH1A1 (0.41) MCHR1ALDH1A1TP53MC4ROPRM1
SCHEMBL27685002 0.82 MCHR1 (0.39) MCHR1ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL27685121 0.80 PSIP1 (0.39) MCHR1ALDH1A1TP53OPRM1OPRD1
SCHEMBL2821958 0.80 FABP3 (0.43) MCHR1ALDH1A1FABP3FABP4PRNP
SCHEMBL27685274 0.78 HSD11B1 (0.36) MCHR1ALDH1A1
SCHEMBL2825540 0.76 ALDH1A1 (0.39) MCHR1ALDH1A1FABP3FABP4PRNP
SCHEMBL27685000 0.74 PSIP1 (0.40) MCHR1ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL27704121 0.71 IDO1 (0.43) ALDH1A1TP53CASP3MAPT
SCHEMBL27685273 0.71 PSIP1 (0.37) MCHR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-A1 QUINOLINE AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS F. Hoffmann-Roche AG (CH) 2007-07-25 EP disclosed
WO-2006048146-A1 QUINOLINE AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-11 WO disclosed