SCHEMBL5240256

SCHEMBL5240256

CS(=O)(=O)c1c[c]ccc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.46
ACLY P53396 1/20 0.38
LOXL2 Q9Y4K0 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAOA P21397 1/20 0.37
LOX P28300 1/20 0.37
PTGS1 P23219 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10709066 0.82 TSHR (0.38) PTGS2KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7366015 0.82 CA2 (0.41) PTGS2CYP2C9PTGS1
SCHEMBL21408564 0.81 GSTO1 (0.44) PTGS2ALDH1A1LMNAHTTKMT2A
SCHEMBL16719623 0.81 SLC22A12 (0.42) PTGS2ACLYPTGS1
SCHEMBL16719861 0.81 PTGS2 (0.39) PTGS2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL207671 0.78 PTGS2 (0.44) PTGS2ACLYKDM4EALDH1A1LMNA
SCHEMBL15703721 0.77 PTGS2 (0.41) PTGS2ACLYKDM4EALDH1A1LMNA
SCHEMBL29415408 0.77 PTGS2 (0.61) PTGS2ACLYKDM4EALDH1A1KMT2A
SCHEMBL937206 0.77 PTGS2 (0.61) PTGS2ACLYKDM4EALDH1A1KMT2A
SCHEMBL2447766 0.75 PTGS2 (0.64) PTGS2ACLYLOXL2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565436-A4 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORP (US) 2007-07-18 EP claimed
JP-2006516145-A 2006-06-22 JP claimed
EP-1565436-A2 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORPORATION (US) 2005-08-24 EP claimed
WO-2004050024-A2 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORPORATION (US) 2004-06-17 WO claimed
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed