SCHEMBL5240356

SCHEMBL5240356

CC(C)Oc1ccccc1N1CCN(C(N)C(C)O)CC1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 6/20 0.52
ADRA1A P35348 6/20 0.52
ADRA1B P35368 5/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7690863 0.85 ADRA1A (0.57) ADRA1DADRA1AADRA1B
Bromide SCHEMBL7683252 0.84 ADRA1A (0.56) ADRA1DADRA1AADRA1B
SCHEMBL6193262 0.81 ADRA1A (0.55) ADRA1DADRA1AADRA1B
SCHEMBL4538062 0.77 ADRA1D (0.58) ADRA1DADRA1AADRA1B
SCHEMBL14621895 0.77 DRD2 (0.67) ADRA1DADRA1AADRA1B
SCHEMBL7301761 0.77 ADRA1A (0.60) ADRA1DADRA1AADRA1B
SCHEMBL3954997 0.76 ADRA1D (0.58) ADRA1DADRA1AADRA1B
SCHEMBL3955000 0.76 ADRA1D (0.58) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL6194198 0.74 ADRA1D (0.52) ADRA1DADRA1AADRA1B
SCHEMBL1050135 0.73 DRD2 (0.60)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758583-A2 ARYLPIPERAZINE DERIVATIVES USEFUL AS ADRENERGIC RECEPTOR ANTAGONISTS Ranbaxy Laboratories Limited (IN) 2007-03-07 EP disclosed
WO-2005118537-A2 ARYLPIPERAZINE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2005-12-15 WO disclosed