SCHEMBL5240728

SCHEMBL5240728

NN=C(Cc1ccnc2ccccc12)c1cccc(C(F)(F)F)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
AURKA O14965 2/20 0.39
AURKB Q96GD4 2/20 0.39
CNR2 P34972 1/20 0.36
KDR P35968 3/20 0.35
KAT6A Q92794 1/20 0.34
RPS6KB1 P23443 1/20 0.34
RIPK1 Q13546 1/20 0.34
CD38 P28907 1/20 0.34
CTSS P25774 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
FLT1 P17948 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
HIF1A Q16665 1/20 0.33
FERMT2 Q96AC1 1/20 0.33
NCF1 P14598 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240723 1.00 CYP1A2 (0.40) CYP1A2LOXL2AURKAAURKBCNR2
SCHEMBL5235891 0.82 CYP1A2 (0.45) CYP1A2LOXL2AURKAAURKBCNR2
SCHEMBL5232563 0.82 LOXL2 (0.46) CYP1A2LOXL2ADORA2AADORA1CYP3A4
SCHEMBL5232556 0.82 LOXL2 (0.46) CYP1A2LOXL2ADORA2AADORA1CYP3A4
SCHEMBL5239698 0.79 KDR (0.38) CYP1A2AURKAAURKBKDRTRPV1
SCHEMBL5235015 0.76 LOXL2 (0.43) CYP1A2LOXL2AURKAAURKBCNR2
SCHEMBL5237502 0.76 LOXL2 (0.43) CYP1A2LOXL2AURKAAURKBCNR2
SCHEMBL27517280 0.76 MEN1 (0.53) CYP1A2CNR2KAT6ACTSSADORA2A
SCHEMBL5231738 0.76 CNR2 (0.45) CYP1A2LOXL2CNR2KDRFLT1
SCHEMBL5240093 0.76 CNR2 (0.45) CYP1A2LOXL2CNR2KDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed