SCHEMBL5235891

SCHEMBL5235891

O=C(Cc1ccnc2ccccc12)c1cccc(C(F)(F)F)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CNR2 P34972 2/20 0.43
AURKA O14965 2/20 0.42
AURKB Q96GD4 2/20 0.42
CTNNB1 P35222 3/20 0.41
WNT3A P56704 3/20 0.41
CTSS P25774 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.39
KAT6A Q92794 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
NSD2 O96028 1/20 0.38
RPS6KB1 P23443 1/20 0.38
CD38 P28907 1/20 0.38
KDR P35968 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240723 0.82 CYP1A2 (0.40) CYP1A2CNR2AURKAAURKBCTSS
SCHEMBL5240728 0.82 CYP1A2 (0.40) CYP1A2CNR2AURKAAURKBCTSS
SCHEMBL5236277 0.80 CYP1A2 (0.52) CYP1A2CTNNB1WNT3ALOXL2KAT6A
SCHEMBL5239743 0.77 VNN1 (0.44) CYP1A2LOXL2RPS6KB1KDRGPBAR1
SCHEMBL5239698 0.76 KDR (0.38) CYP1A2AURKAAURKBTRPV1KDR
SCHEMBL5239397 0.74 CNR2 (0.50) CYP1A2CNR2LOXL2KDR
SCHEMBL5239399 0.74 CYP1A2 (0.46) CYP1A2LOXL2ADORA2AADORA1
SCHEMBL5233508 0.74 CNR2 (0.53) CYP1A2CNR2KDR
Bromide SCHEMBL5257264 0.74 CYP1A2 (0.51) CYP1A2CTNNB1WNT3ALOXL2NSD2
SCHEMBL5237313 0.72 RAB9A (0.56) CYP1A2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed