SCHEMBL5240809

SCHEMBL5240809

[CH2]c1nn(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)c1Cc1cccc(OC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADCY10 Q96PN6 1/20 0.39
FPR1 P21462 3/20 0.38
FPR2 P25090 2/20 0.38
TAAR1 Q96RJ0 2/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
IDH1 O75874 1/20 0.35
PPARG P37231 1/20 0.35
LTA4H P09960 1/20 0.35
DHFR P00374 1/20 0.35
CCNB2 O95067 1/20 0.35
CCNE2 O96020 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
PDE1B Q01064 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240819 0.89 MEN1 (0.41) ADCY10FPR1FPR2TAAR1LMNA
SCHEMBL5214219 0.87 FPR1 (0.39) ADCY10FPR1FPR2TAAR1LMNA
SCHEMBL5244652 0.81 FLT1 (0.34) ALDH1A1
SCHEMBL5244481 0.77 CYP1A2 (0.33) HTR6POLB
SCHEMBL5239631 0.76 ADCY10 (0.39) ADCY10LMNAMAPTCDK4CCND1
SCHEMBL5640684 0.74 ALDH1A1 (0.38) ADCY10LMNAMAPTPDE1BPDE1C
SCHEMBL5239947 0.73 GRM5 (0.32)
SCHEMBL5643053 0.73 ENPP1 (0.35) ADCY10POLB
SCHEMBL5243348 0.73 CNR1 (0.33)
SCHEMBL5640193 0.71 PDE1A (0.35) PDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401826-B1 PYRAZOLE DERIVATIVES AS HIV REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP claimed