SCHEMBL5243158

SCHEMBL5243158

CCCCCC(N1CCN(c2cccc(Cl)c2)CC1)N1CCN(c2cccc(Cl)c2)CC1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
LMNA P02545 2/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
RECQL P46063 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
ALOX12 P18054 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5243181 0.85 KCNH2 (0.54) KCNH2MAPK1ALDH1A1MAPT
SCHEMBL5247341 0.83 DRD2 (0.51) KCNH2LMNATSHRNPSR1ALDH1A1
SCHEMBL5244521 0.83 DRD2 (0.59) KCNH2TSHRALDH1A1MAPTSMN1; SMN2
SCHEMBL8128745 0.81 HTR3E (0.53) KCNH2HTR3EHTR3BHTR3AHTR3D
SCHEMBL13875118 0.79 KCNH2 (0.83) KCNH2
SCHEMBL2214111 0.78 KCNH2 (0.86) KCNH2
SCHEMBL10414971 0.77 KCNH2 (0.80) KCNH2
SCHEMBL7835678 0.76 LMNA (0.49) KCNH2LMNATSHRMAPK1RECQL
SCHEMBL11955707 0.76 HTR3E (0.58) KCNH2LMNATSHRNPSR1HTR3E
Hydrochloric Acid SCHEMBL10372885 0.76 LMNA (0.54) KCNH2LMNATSHRMAPK1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836192-A2 ARYL PIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS Universita' Degli Studi di Siena (IT) 2007-09-26 EP claimed
WO-2006072608-A2 ARYL PIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS UNIVERSITÁ DEGLI STUDI DI SIENA (IT) 2006-07-13 WO claimed
EP-1836192-A2 ARYL PIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS Universita' Degli Studi di Siena (IT) 2007-09-26 EP disclosed
WO-2006072608-A2 ARYL PIPERAZINE DERIVATIVES FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS UNIVERSITÁ DEGLI STUDI DI SIENA (IT) 2006-07-13 WO disclosed