SCHEMBL5244207

SCHEMBL5244207

O=C(O)N1CCc2sc(S(=O)(=O)Nc3ccccc3NS(=O)(=O)c3cc4ccccc4s3)cc2C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.45
MCL1 Q07820 1/20 0.43
HDAC1 Q13547 1/20 0.41
MMP13 P45452 1/20 0.40
F10 P00742 1/20 0.40
GHSR Q92847 1/20 0.38
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
RECQL P46063 1/20 0.37
CA2 P00918 1/20 0.36
HTT P42858 2/20 0.36
PLA2G1B P04054 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PKM P14618 1/20 0.35
ACLY P53396 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192421 0.86 MMP13 (0.53) CCR2MCL1HDAC1MMP13F10
SCHEMBL5244220 0.83 MMP13 (0.39) CCR2MCL1HDAC1MMP13F10
SCHEMBL4188720 0.76 CCR2 (0.64) CCR2MCL1HDAC1GHSRCA2
SCHEMBL4192431 0.73 MMP13 (0.51) MMP13F10HDAC6
SCHEMBL2689511 0.72 CCR2 (0.54) CCR2MCL1HDAC1LMNACA2
SCHEMBL28769697 0.72 HDAC6 (0.40) F10LMNACA2NPC1RAB9A
SCHEMBL21999998 0.71 ACLY (0.55) MCL1ACLY
SCHEMBL10143420 0.70 CCR2 (0.57) CCR2MCL1HDAC1F10GHSR
SCHEMBL10238662 0.70 CCR2 (0.45) CCR2MCL1HDAC1MMP13GHSR
Hydrochloric Acid SCHEMBL9958452 0.69 CCR2 (0.44) CCR2MCL1HDAC1MMP13GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809619-A1 BISSULFONAMIDE COMPOUNDS AS AGONISTS OF GALR1, COMPOSITIONS, AND METHODS OF USE Transtech Pharma, Inc. (US) 2007-07-25 EP disclosed
WO-2006047302-A1 BISSULFONAMIDE COMPOUNDS AS AGONISTS OF GALR1, COMPOSITIONS, AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2006-05-04 WO disclosed