SCHEMBL5244706

SCHEMBL5244706

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3cc(F)cc(F)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.40
ROCK1 Q13464 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
BRD4 O60885 5/20 0.38
MIF P14174 2/20 0.37
PDE10A Q9Y233 1/20 0.36
DDT P30046 3/20 0.36
HTR7 P34969 1/20 0.36
AURKA O14965 1/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244462 0.94 MAPT (0.40) BRD4MIFTP53THRB
SCHEMBL5244376 0.94 PSEN1 (0.41) ROCK2ROCK1EGLN1DDTPSEN1
SCHEMBL5246709 0.94 ROCK2 (0.42) ROCK2ROCK1BRD4MIFPDE10A
SCHEMBL5246767 0.92 MIF (0.47) BRD4MIFDDTPSEN1PSEN2
SCHEMBL5245935 0.91 ROCK2 (0.41) ROCK2ROCK1BRD4MIFPDE10A
SCHEMBL5245221 0.90 HPGD (0.44) BRD4DDTPSEN1PSEN2APH1B
SCHEMBL5248109 0.90 EGLN1 (0.38) ROCK2ROCK1EGLN1MIFPDE10A
SCHEMBL5244638 0.89 LMNA (0.39) ROCK2ROCK1BRD4DDT
SCHEMBL5247657 0.89 LMNA (0.46) BRD4MIFDDT
SCHEMBL5245898 0.89 PPARG (0.40) ROCK2ROCK1BRD4PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed