SCHEMBL5247657

SCHEMBL5247657

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3ccc(Cl)c(Cl)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
IKBKB O14920 1/20 0.39
MAOB P27338 1/20 0.38
EPHX2 P34913 1/20 0.37
PPARG P37231 1/20 0.37
WDR5 P61964 3/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
BRD4 O60885 1/20 0.36
NOTUM Q6P988 1/20 0.36
DDT P30046 1/20 0.36
CXCR3 P49682 1/20 0.36
MIF P14174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244638 0.94 LMNA (0.39) LMNAWDR5BRD4DDT
SCHEMBL5245570 0.91 LMNA (0.42) LMNAMAOBEPHX2WDR5HDAC4
SCHEMBL5246245 0.90 ROCK2 (0.41) BRD4DDTMIF
SCHEMBL5245935 0.90 ROCK2 (0.41) BRD4DDTMIF
SCHEMBL5244462 0.90 MAPT (0.40) BRD4MIF
SCHEMBL5244706 0.89 ROCK2 (0.40) BRD4DDTMIF
SCHEMBL5246767 0.89 MIF (0.47) LMNAEPHX2BRD4DDTMIF
SCHEMBL5246709 0.88 ROCK2 (0.42) LMNABRD4DDTMIF
SCHEMBL5247395 0.88 DDT (0.43) EPHX2PPARGHDAC1DDTMIF
SCHEMBL5247966 0.88 EPHX2 (0.43) LMNAEPHX2HDAC8HDAC6MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed