SCHEMBL5246018

SCHEMBL5246018

C=CCCCOc1cc(C(=O)NCC)ccc1-n1cc(C(=O)NCc2cccc(F)c2)nn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
GLS O94925 1/20 0.41
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 1/20 0.41
DDT P30046 3/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
CNR1 P21554 1/20 0.39
MMP13 P45452 1/20 0.39
BRD4 O60885 2/20 0.39
PSEN1 P49768 2/20 0.39
PSEN2 P49810 2/20 0.39
APH1B Q8WW43 2/20 0.39
NCSTN Q92542 2/20 0.39
APH1A Q96BI3 2/20 0.39
PSENEN Q9NZ42 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
PDE10A Q9Y233 1/20 0.38
MIF P14174 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5245598 0.91 GLS (0.44) POLBGLSROCK2ROCK1DDT
SCHEMBL5247632 0.89 GLS (0.42) POLBGLSROCK2ROCK1DDT
SCHEMBL5246709 0.88 ROCK2 (0.42) POLBGLSROCK2ROCK1DDT
SCHEMBL5244275 0.85 MAPK8 (0.47)
SCHEMBL5248477 0.85 BRD4 (0.47) POLBMAPTBRD4TP53
SCHEMBL5243944 0.84 SMPD1 (0.39) BRD4TP53
SCHEMBL5247498 0.83 SMPD1 (0.39) POLBBRD4TP53
SCHEMBL5244405 0.83 KMT2A (0.38) MAPTBRD4LMNATP53
SCHEMBL5244829 0.83 BRD4 (0.37) BRD4TP53
SCHEMBL5244377 0.83 BRD4 (0.38) BRD4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed