SCHEMBL5246364

SCHEMBL5246364

N#Cc1cccc([S+]([O-])N2CCN(c3ccccc3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.51
DRD3 P35462 6/20 0.51
NOTUM Q6P988 1/20 0.45
SLC2A1 P11166 1/20 0.43
SLC2A2 P11168 1/20 0.43
SLC2A3 P11169 1/20 0.43
DRD4 P21917 4/20 0.42
HTR1A P08908 1/20 0.42
C1S P09871 1/20 0.41
DHFR P00374 2/20 0.40
POLB P06746 1/20 0.40
MLYCD O95822 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
CHRM4 P08173 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5243882 0.85 POLB (0.48) DRD2DRD3DRD4HTR1APOLB
SCHEMBL18581653 0.83 DRD2 (0.41) DRD2DRD3NOTUM
SCHEMBL20195330 0.83 DRD2 (0.41) DRD2DRD3NOTUM
SCHEMBL5244482 0.81 ALDH1A1 (0.44) DRD2DRD4HTR1APOLB
SCHEMBL15800697 0.77 DRD2 (0.79) DRD2DRD3NOTUMSLC2A1SLC2A2
SCHEMBL5247322 0.73 DRD2 (0.42) DRD2DRD3DRD4HTR1APOLB
SCHEMBL3537217 0.71 DRD2 (0.74) DRD2DRD3NOTUMSLC2A1SLC2A2
SCHEMBL29809089 0.71 DRD2 (0.74) DRD2DRD3NOTUMSLC2A1SLC2A2
SCHEMBL22495307 0.71 DRD2 (0.64) DRD2DRD3NOTUMSLC2A1SLC2A2
SCHEMBL5245726 0.70 LMNA (0.54) DRD2DRD3DRD4HTR1APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866298-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2007-12-19 EP claimed
WO-2006105127-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-10-05 WO claimed