SCHEMBL5247166

SCHEMBL5247166

CC(C)(C)c1ccc(CNC(=O)c2cn(-c3ccc(C(=O)NCC(F)(F)F)cc3OCCOCCF)nn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 13/20 0.41
NR1H4 Q96RI1 11/20 0.41
DDT P30046 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
MIF P14174 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246995 0.94 DDT (0.41) EPHX2DDTMIF
SCHEMBL5247966 0.92 EPHX2 (0.43) EPHX2NR1H4MEN1KMT2ANPC1
SCHEMBL5246077 0.92 MMP13 (0.37) EPHX2DDTHDAC8MIF
SCHEMBL5246041 0.91 MIF (0.45) EPHX2DDTMIF
SCHEMBL5244132 0.89 HTR2C (0.43) EPHX2NR1H4CYP1A2CYP2C19
SCHEMBL5246799 0.89 PSEN1 (0.41) DDTCYP1A2CYP2C19MIF
SCHEMBL5248109 0.89 EGLN1 (0.38) EPHX2DDTHDAC8MIF
SCHEMBL5247824 0.89 MMP13 (0.39) EPHX2DDTMIF
SCHEMBL5245570 0.88 LMNA (0.42) EPHX2DDTHDAC8HDAC6
SCHEMBL5247395 0.88 DDT (0.43) EPHX2DDTMIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed