SCHEMBL5247302

SCHEMBL5247302

Cc1onc(-c2ccccc2Cl)c1OC(=O)O.Cc1sc(-c2ccccc2)nc1CC(=O)NC1CCC(Cc2ccccc2)(N(C)C)CC1.Cc1sc(-c2ccccc2)nc1CC(=O)NC1CCC(Cc2ccccc2F)(N(C)C)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
PPARG P37231 2/20 0.35
NCOA2 Q15596 2/20 0.35
KMT2A Q03164 4/20 0.35
LMNA P02545 4/20 0.35
ALDH1A1 P00352 4/20 0.35
MEN1 O00255 2/20 0.35
HTT P42858 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
GABRA5 P31644 3/20 0.34
MAPT P10636 2/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5245606 0.89 KMT2A (0.38) KDM4EPPARGNCOA2KMT2ALMNA
SCHEMBL316431 0.83 KMT2A (0.42) PPARGKMT2ALMNAALDH1A1MEN1
SCHEMBL5245278 0.81 KMT2A (0.33) KMT2ALMNAALDH1A1MEN1HTT
SCHEMBL5245600 0.79 KMT2A (0.44) KDM4EPPARGNCOA2KMT2ALMNA
SCHEMBL316821 0.78 OPRM1 (0.46) PPARGKMT2ALMNAALDH1A1MEN1
SCHEMBL315932 0.76 LMNA (0.41) KDM4EPPARGKMT2ALMNAALDH1A1
SCHEMBL316610 0.76 OPRM1 (0.41) PPARGKMT2ALMNAALDH1A1MEN1
SCHEMBL315482 0.75 KMT2A (0.62) KMT2ALMNAALDH1A1MEN1HTT
SCHEMBL315905 0.74 SIGMAR1 (0.43) PPARGKMT2ALMNAMEN1MAPT
SCHEMBL315989 0.71 OPRM1 (0.44) PPARGKMT2ALMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745009-A1 HETEROARYL SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP disclosed
WO-2005110971-A1 HETEROARYL SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO disclosed