SCHEMBL5247939

SCHEMBL5247939

CCOC(=O)N1C2CCC1CC(O)(c1ccc(Cl)c(OC)c1)C2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.47
BRAF P15056 1/20 0.45
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
CHRM1 P11229 2/20 0.39
POLB P06746 2/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
HTT P42858 3/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14081574 0.77 GRM5 (0.53) GRM5ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL5905121 0.76 DRD2 (0.52)
SCHEMBL5194325 0.75 DRD2 (0.48) ALDH1A1
SCHEMBL5193723 0.74 DRD2 (0.48)
SCHEMBL5798011 0.74 DRD2 (0.43)
SCHEMBL5195811 0.73 DRD2 (0.40) ALDH1A1SMN1; SMN2
SCHEMBL5798010 0.72 OPRM1 (0.43)
SCHEMBL5196784 0.72 HTR4 (0.36) BRAFSMN1; SMN2MAPTMAPK1
SCHEMBL5194165 0.71 DRD2 (0.40) ALDH1A1SMN1; SMN2
SCHEMBL5905435 0.70 DRD2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809626-A2 ARYL SUBSTITUTED 8-AZABICYCLO[3.2.1]OCTANE COMPOUNDS AS LIGANDS OF THE MELANIN CONCENTRATING HORMONE RECEPTOR Neurogen Corporation (US) 2007-07-25 EP disclosed
WO-2006044174-A9 ARYL SUBSTITUTED 8-AZABICYCLO[3.2.1]OCTANE COMPOUNDS AS LIGANDS OF THE MELANIN CONCENTRATING HORMONE RECEPTOR NEUROGEN CORP (US) 2006-07-20 WO disclosed
WO-2006044174-A2 ARYL SUBSTITUTED 8-AZABICYCLO[3.2.1]OCTANE COMPOUNDS AS LIGANDS OF THE MELANIN CONCENTRATING HORMONE RECEPTOR NEUROGEN CORPORATION (US) 2006-04-27 WO disclosed