SCHEMBL5250855

SCHEMBL5250855

O=c1[nH]cc([N+](=O)[O-])c(Cl)c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44
GLA P06280 1/20 0.44
GPR35 Q9HC97 1/20 0.39
RAB9A P51151 1/20 0.39
TSHR P16473 4/20 0.37
GRIN2D O15399 3/20 0.37
GRIN3B O60391 3/20 0.37
GRIN1 Q05586 3/20 0.37
GRIN2A Q12879 3/20 0.37
GRIN2B Q13224 3/20 0.37
GRIN2C Q14957 3/20 0.37
GRIN3A Q8TCU5 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
HPGD P15428 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
GRIK1 P39086 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13458098 0.81 ALDH1A1 (0.33) ALDH1A1KDM4EGLA
SCHEMBL1200250 0.78 KDM4E (0.53) ALDH1A1KDM4EGLAGPR35RAB9A
SCHEMBL9124172 0.74 GPR35 (0.45) ALDH1A1KDM4EGPR35RAB9ATSHR
SCHEMBL3214901 0.70 ALDH1A1 (0.49) ALDH1A1KDM4EGLATSHRGRIN2D
SCHEMBL9860083 0.70 TDP1 (0.59) ALDH1A1GPR35TSHRCYP1A2CYP3A4
SCHEMBL173688 0.69 KDM4E (0.61) ALDH1A1KDM4EGLAGPR35RAB9A
SCHEMBL458846 0.69 KDM4E (0.61) ALDH1A1KDM4EGLAGPR35RAB9A
SCHEMBL29071029 0.68 DNA2 (0.37) ALDH1A1KDM4EGLAGPR35RAB9A
SCHEMBL30449050 0.68 DNA2 (0.37) ALDH1A1KDM4EGLAGPR35RAB9A
SCHEMBL28825088 0.67 GPR35 (0.52) ALDH1A1GPR35TSHRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100056535-A1 Inhibitors of HIV-1 reverse transcriptase ROCHE PALO ALTO LLC 2010-03-04 US disclosed
EP-1670466-A4 PREPARATION OF 1, 6, 7- TRISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LTD (GB) 2007-04-25 EP disclosed
US-20070004771-A1 Preparation of 1,6,7-trisubstituted azabenzimidazoles as kinase inhibitors GLAXO GROUP LIMITED 2007-01-04 US disclosed
EP-1670466-A2 PREPARATION OF 1, 6, 7- TRISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-06-21 EP disclosed
WO-2005034866-A2 PREPARATION OF 1, 6, 7- TRISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056535-A1 Inhibitors of HIV-1 reverse transcriptase QTRT1, NQO2, QTRT2 ALDH1A1 301/4885KDM4E 750/4885GLA 1551/4885
US-20070004771-A1 Preparation of 1,6,7-trisubstituted azabenzimidazoles as kinase inhibitors ROCK1, TNK2, ARHGDIB ALDH1A1 4385/4885KDM4E 969/4885GLA 3710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.