SCHEMBL5253147

SCHEMBL5253147

CCOc1ccnc(N2CCN(C(=O)c3sccc3C#N)CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
RIPK1 Q13546 1/20 0.40
ALDH1A1 P00352 5/20 0.39
KDR P35968 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
SLC6A7 Q99884 2/20 0.39
HPGD P15428 1/20 0.39
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5307963 0.99 LMNA (0.40) LMNARIPK1ALDH1A1KDRCA12
SCHEMBL5254259 0.92 RIPK1 (0.39) LMNARIPK1ALDH1A1KDRCA12
Hydrochloric Acid SCHEMBL5251801 0.92 RIPK1 (0.38) LMNARIPK1ALDH1A1KDRCA12
SCHEMBL5250616 0.92 HRH2 (0.39) LMNARIPK1ALDH1A1KDRCA12
SCHEMBL5254333 0.90 ALDH1A1 (0.44) ALDH1A1KDRSLC6A7HPGDHCRTR1
Hydrochloric Acid SCHEMBL5252156 0.89 ALDH1A1 (0.43) ALDH1A1KDRSLC6A7HPGDHCRTR1
SCHEMBL6651929 0.85 HRH2 (0.44) LMNAALDH1A1CA12CA1CA2
Hypochlorous Acid SCHEMBL6657831 0.84 HRH2 (0.43) LMNAALDH1A1CA12CA1CA2
Hydrochloric Acid SCHEMBL6657823 0.84 HRH2 (0.43) LMNAALDH1A1CA12CA1CA2
SCHEMBL5251523 0.82 HCRTR1 (0.50) LMNAALDH1A1SLC6A7HPGDHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327630-B1 NEW DERIVATIVES OF CYANO-ARYL (OR CYANOHETEROARYL)-CARBONYL-PIPERAZINYL-PYRIMIDINES, THEIR PREPARATION AND APPLICATION AS MEDICATION ESTEVE LABOR DR (ES) 2007-12-12 EP claimed
US-7300937-B2 Derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl-pyrimidines, their preparation and application as medication LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-11-27 US claimed
EP-1327630-A1 NEW DERIVATIVES OF CYANO-ARYL (OR CYANOHETEROARYL)-CARBONYL-PIPERAZINYL-PYRIMIDINES, THEIR PREPARATION AND APPLICATION AS MEDICATION LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2003-07-16 EP claimed