SCHEMBL5254259

SCHEMBL5254259

CCCOc1ccnc(N2CCN(C(=O)c3sccc3C#N)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.39
ACACB O00763 1/20 0.39
ALDH1A1 P00352 4/20 0.38
KDR P35968 1/20 0.38
SLC6A7 Q99884 4/20 0.37
HPGD P15428 1/20 0.37
KDM4E B2RXH2 5/20 0.37
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PANK3 Q9H999 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5251801 0.99 RIPK1 (0.38) RIPK1ACACBALDH1A1KDRSLC6A7
SCHEMBL5250616 0.95 HRH2 (0.39) RIPK1ACACBALDH1A1KDRSLC6A7
SCHEMBL5253147 0.92 LMNA (0.41) RIPK1ALDH1A1KDRSLC6A7HPGD
Hydrochloric Acid SCHEMBL5307963 0.91 LMNA (0.40) RIPK1ALDH1A1KDRSLC6A7HPGD
SCHEMBL5254333 0.88 ALDH1A1 (0.44) ALDH1A1KDRSLC6A7HPGDKDM4E
Hydrochloric Acid SCHEMBL5252156 0.87 ALDH1A1 (0.43) ALDH1A1KDRSLC6A7HPGDKDM4E
SCHEMBL5254634 0.83 GBA1 (0.47) ALDH1A1SLC6A7HPGDKDM4ELMNA
SCHEMBL5251934 0.82 KDM4E (0.44) ACACBALDH1A1SLC6A7HPGDKDM4E
Hydrochloric Acid SCHEMBL5255413 0.82 GBA1 (0.46) ALDH1A1SLC6A7HPGDKDM4ELMNA
Hydrochloric Acid SCHEMBL5253011 0.81 KDM4E (0.43) ACACBALDH1A1SLC6A7HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327630-B1 NEW DERIVATIVES OF CYANO-ARYL (OR CYANOHETEROARYL)-CARBONYL-PIPERAZINYL-PYRIMIDINES, THEIR PREPARATION AND APPLICATION AS MEDICATION ESTEVE LABOR DR (ES) 2007-12-12 EP claimed
US-7300937-B2 Derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl-pyrimidines, their preparation and application as medication LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-11-27 US claimed
EP-1327630-A1 NEW DERIVATIVES OF CYANO-ARYL (OR CYANOHETEROARYL)-CARBONYL-PIPERAZINYL-PYRIMIDINES, THEIR PREPARATION AND APPLICATION AS MEDICATION LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2003-07-16 EP claimed