SCHEMBL5253996

SCHEMBL5253996

C=CCONC1CN(C(=O)O)Cc2nc(NC(C)=O)ncc21

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.33
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
HTR1F P30939 1/20 0.33
MAPK1 P28482 2/20 0.33
SHMT2 P34897 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
SYK P43405 1/20 0.31
CCNK O75909 1/20 0.30
CDK12 Q9NYV4 1/20 0.30
EGFR P00533 1/20 0.30
JAK3 P52333 1/20 0.30
ITK Q08881 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5186351 0.79 TP53 (0.37) TP53HTR1AHTR1DHTR1BHTR1F
SCHEMBL5255776 0.76 HSD11B1 (0.32)
SCHEMBL5255401 0.74
SCHEMBL5257162 0.72
SCHEMBL5254049 0.70
SCHEMBL5253467 0.69 ALDH1A1 (0.33)
SCHEMBL4696280 0.69 NPC1 (0.41)
SCHEMBL5254555 0.68
SCHEMBL18209780 0.67 LMNA (0.31)
SCHEMBL5225649 0.65 POLB (0.38) CCNKCDK12JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed