SCHEMBL5254100

SCHEMBL5254100

COc1cccc2c([C@@H](O)CN3CCC(NC(C4=CC=CCC4)C4=COC=CO4)CC3)ccnc12

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.36
SLC2A1 P11166 12/20 0.35
SIGMAR1 Q99720 1/20 0.33
ABCB1 P08183 2/20 0.31
KCNJ1 P48048 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3686883 0.96 KCNH2 (0.34) KCNH2SLC2A1SIGMAR1
SCHEMBL5262026 0.89 KCNH2 (0.32) KCNH2
SCHEMBL3697776 0.88 SLC2A1 (0.38) KCNH2SLC2A1SIGMAR1ABCB1
SCHEMBL5255791 0.85 KCNH2 (0.52) KCNH2SLC2A1
SCHEMBL3695685 0.84 DRD4 (0.30)
SCHEMBL5254382 0.84 KCNH2 (0.51) KCNH2SLC2A1
SCHEMBL3775157 0.83 KCNH2 (0.41) KCNH2SLC2A1
SCHEMBL3694994 0.83
SCHEMBL3694128 0.82 HTR1A (0.32)
SCHEMBL5650870 0.81 KCNH2 (0.49) KCNH2SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359908-B1 QUINOLINES AND NITROGENATED DERIVATIVES THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2007-08-22 EP claimed