SCHEMBL5254567

SCHEMBL5254567

CS(=O)(=O)O[C@@H]1CN(C(=O)O)[C@H](C(=O)O)c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACE P12821 11/20 0.36
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
FFAR2 O15552 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187913 0.88 MMP2 (0.36)
SCHEMBL5260323 0.73 ACE (0.42) ACEPOLB
SCHEMBL5256022 0.72 ACE (0.41) ACEPOLB
SCHEMBL19470993 0.68 DRD1 (0.57) CYP3A4
SCHEMBL17674610 0.68 DRD1 (0.57) CYP3A4
SCHEMBL5254943 0.66 NPC1 (0.38) ACEL3MBTL1
SCHEMBL5023851 0.65 ACE (0.66) ACE
SCHEMBL5185349 0.65 MMP2 (0.40) POLB
SCHEMBL5253676 0.64 ACE (0.36) ACEPOLBCYP3A4
SCHEMBL5257429 0.64 ALDH1A1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed