SCHEMBL5255129

SCHEMBL5255129

Cc1ccc2c(c1)N(C1CCN(C(=O)OC(C)(C)C)CC1)CC2

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
GPR119 Q8TDV5 3/20 0.51
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
ALOX12 P18054 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ESR2 Q92731 1/20 0.46
NR1H2 P55055 1/20 0.46
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
EPHX2 P34913 1/20 0.45
MEN1 O00255 1/20 0.43
KDM4E B2RXH2 1/20 0.43
THRB P10828 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN6 P29350 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5254230 0.91 TP53 (0.53) TP53GPR119NPC1RAB9AKMT2A
SCHEMBL15009205 0.87 HTR1A (0.50)
SCHEMBL5871429 0.87 FPR2 (0.51) TP53GPR119NPC1RAB9AESR2
SCHEMBL4993502 0.87 ESR2 (0.48) TP53GPR119NPC1RAB9AKMT2A
SCHEMBL5871267 0.85 TP53 (0.50) TP53GPR119NPC1RAB9AESR2
SCHEMBL5870923 0.84 TP53 (0.49) TP53GPR119NPC1RAB9AESR2
SCHEMBL12459066 0.84 ALDH1A1 (0.53) TP53GPR119NPC1RAB9AESR2
SCHEMBL2707784 0.84 GPR119 (0.52) TP53GPR119NPC1RAB9AKDM4E
SCHEMBL4114089 0.81 NR1H2 (0.59) TP53GPR119NPC1RAB9AESR2
SCHEMBL2774721 0.81 SMN1; SMN2 (0.49) TP53GPR119KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed