SCHEMBL5255287

SCHEMBL5255287

CC(C)CN(CC(C)C)S(=O)(=O)N[C@@](C)(Cc1ccc(Nc2nccc3cnccc23)cc1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
TRPV1 Q8NER1 5/20 0.33
ADRB3 P13945 4/20 0.32
MMP1 P03956 1/20 0.31
ADAM17 P78536 1/20 0.31
NAMPT P43490 1/20 0.30
P2RX3 P56373 1/20 0.30
P2RX7 Q99572 1/20 0.30
KDR P35968 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5256231 0.90 TRPV1 (0.34) HDAC3HDAC1HDAC6TRPV1ADRB3
SCHEMBL5259963 0.88 ADRB3 (0.37) HDAC3HDAC1HDAC6TRPV1ADRB3
SCHEMBL5257628 0.85 CYP3A4 (0.36) TRPV1P2RX7
SCHEMBL5255321 0.84 JAK3 (0.37) ADRB3NAMPT
SCHEMBL5225642 0.82 ITGB1 (0.36) HDAC3HDAC1HDAC6TRPV1P2RX3
SCHEMBL5255283 0.79 CA12 (0.37) HDAC3HDAC1HDAC6TRPV1P2RX3
SCHEMBL5258338 0.77 NAMPT (0.37) TRPV1ADRB3NAMPT
SCHEMBL5256333 0.75 FFAR1 (0.37) TRPV1P2RX7
SCHEMBL5228649 0.73 ITGB1 (0.37) HDAC3HDAC1HDAC6TRPV1P2RX3
SCHEMBL5264743 0.73 TRPV1 (0.42) HDAC3HDAC1HDAC6TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622867-B1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN ALPHA4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-19 EP claimed
EP-1622867-B1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN ALPHA4 ANTAGONISTS ALMIRALL LAB (ES) 2007-09-19 EP disclosed