SCHEMBL5260586

SCHEMBL5260586

CCCCN(C=O)c1c[nH]c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
BCHE P06276 3/20 0.44
MAPT P10636 5/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
RAB9A P51151 2/20 0.44
MITF O75030 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB2 P47870 1/20 0.44
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
HTR2A P28223 2/20 0.43
CYP2A6 P11509 1/20 0.42
IMPDH2 P12268 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6608825 0.82 NPC1 (0.41) NPC1SMN1; SMN2BCHEMAPTMEN1
SCHEMBL5792372 0.79 NPC1 (0.46) NPC1SMN1; SMN2BCHEMAPTMEN1
SCHEMBL14399666 0.74 HTR2A (0.53) NPC1MAPTMEN1KMT2AALDH1A1
SCHEMBL5010711 0.74 HTR1B (0.46) SMN1; SMN2BCHEMEN1KMT2AALDH1A1
SCHEMBL6608957 0.73 NPC1 (0.42) NPC1SMN1; SMN2BCHEMAPTMEN1
SCHEMBL27407793 0.71 IMPDH2 (0.50) NPC1MAPTMEN1KMT2AALDH1A1
SCHEMBL7973209 0.71 CYP2A6 (0.50) NPC1MAPTMEN1KMT2AALDH1A1
SCHEMBL4982358 0.71 MEN1 (0.54) NPC1MAPTMEN1KMT2AALDH1A1
SCHEMBL5010601 0.70 HTR1B (0.41) KMT2AALDH1A1TDP1CYP2C9
SCHEMBL17782579 0.70 MC4R (0.57) NPC1SMN1; SMN2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379239-B1 N-(2-ARYLETHYL) BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR LILLY CO ELI (US) 2007-09-12 EP disclosed
EP-1379239-A2 N-(2-ARYLETHYL) BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2004-01-14 EP disclosed
WO-2002078693-A2 N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2002-10-10 WO disclosed