SCHEMBL5261323

SCHEMBL5261323

O=C(NCCCN1CCOCC1)c1cc(Cl)ccc1NC(=O)c1cccc2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.62
BCL3 P20749 2/20 0.60
POLB P06746 1/20 0.60
KMT2A Q03164 2/20 0.58
CNR1 P21554 1/20 0.58
CNR2 P34972 1/20 0.58
ALDH1A1 P00352 3/20 0.56
MEN1 O00255 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
SLC6A4 P31645 1/20 0.55
LMNA P02545 1/20 0.55
KLK7 P49862 1/20 0.54
KDM4E B2RXH2 1/20 0.53
HPGD P15428 1/20 0.53
TSHR P16473 1/20 0.53
MAOA P21397 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258790 0.94 HTT (0.70) HTTBCL3KMT2ACNR1CNR2
SCHEMBL17554125 0.90 BCL3 (0.74) HTTBCL3POLBKMT2AALDH1A1
SCHEMBL4204512 0.85 HTT (0.55) HTTPOLBKMT2ACNR1CNR2
SCHEMBL17554166 0.83 BCL3 (0.73) HTTBCL3POLBKMT2AALDH1A1
SCHEMBL4191608 0.83 CNR1 (0.59) HTTBCL3KMT2ACNR1CNR2
SCHEMBL4195045 0.82 MEN1 (0.57) HTTPOLBKMT2ACNR1CNR2
SCHEMBL5258216 0.81 CNR1 (0.67) HTTKMT2ACNR1CNR2ALDH1A1
SCHEMBL4190787 0.80 CNR1 (0.65) HTTPOLBKMT2ACNR1CNR2
SCHEMBL5795351 0.80 KMT2A (0.63) HTTBCL3KMT2AALDH1A1MEN1
SCHEMBL31518356 0.80 KMT2A (0.63) HTTBCL3KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed