SCHEMBL5263671

SCHEMBL5263671

CC(=O)OOc1cccc(C#N)c1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.38
MAPK1 P28482 1/20 0.38
ACHE P22303 1/20 0.37
ALDH1A1 P00352 6/20 0.37
NOTUM Q6P988 1/20 0.37
TSHR P16473 3/20 0.37
HPGD P15428 1/20 0.37
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
GAA P10253 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAOB P27338 1/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
IMPDH2 P12268 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5970515 0.85 SMN1; SMN2 (0.47) SMN1; SMN2MAPK1ALDH1A1TSHRHPGD
SCHEMBL21728172 0.83 ACHE (0.54) SSTR4SMN1; SMN2MAPK1ACHEALDH1A1
SCHEMBL11139550 0.78 POLB (0.46) ACHEALDH1A1HPGDNPC1RAB9A
SCHEMBL1432109 0.75 KMT2A (0.41) SMN1; SMN2MAPK1ACHEALDH1A1TSHR
SCHEMBL4595414 0.74 ALDH1A1 (0.43) ALDH1A1HPGDNPC1RAB9AGAA
SCHEMBL4119375 0.73 POLB (0.50) SMN1; SMN2ACHEALDH1A1TSHRGAA
SCHEMBL1959471 0.72 ERN1 (0.53) SMN1; SMN2ACHEALDH1A1TSHRHPGD
SCHEMBL22172091 0.72 TSHR (0.43) SSTR4SMN1; SMN2MAPK1ACHEALDH1A1
SCHEMBL30957147 0.71 TSHR (0.44) SSTR4SMN1; SMN2MAPK1ALDH1A1TSHR
SCHEMBL5636872 0.70 TSHR (0.42) SSTR4SMN1; SMN2MAPK1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed