SCHEMBL5266006

SCHEMBL5266006

O=C(CCc1ccccc1)Nc1c[nH]nc1C(=O)NCCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.51
NPC1 O15118 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 2/20 0.48
POLB P06746 2/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48
HTT P42858 2/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK2 O75116 1/20 0.46
KDM6B O15054 1/20 0.45
KDM4D Q6B0I6 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
EGLN3 Q9H6Z9 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267185 0.90 POLB (0.48) RAB9ANPC1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL5266469 0.87 SMN1; SMN2 (0.56) RAB9ANPC1SMN1; SMN2ALDH1A1LMNA
SCHEMBL5272569 0.86 MAPT (0.58) RAB9ANPC1SMN1; SMN2KDM4EPOLB
SCHEMBL5268734 0.86 KDM4E (0.51) RAB9ANPC1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL5268958 0.86 RAB9A (0.52) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL5269503 0.86 RAB9A (0.61) RAB9ANPC1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL5270533 0.85 MEN1 (0.47) RAB9ANPC1SMN1; SMN2ALDH1A1LMNA
SCHEMBL5269224 0.84 KDM4E (0.49) RAB9ANPC1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL13816928 0.84 RAB9A (0.54) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL5269702 0.83 EPHX2 (0.49) RAB9ANPC1SMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed