SCHEMBL5266752

SCHEMBL5266752

O=C(Nc1c[nH]nc1C(=O)Nc1ccccc1)c1ccc(F)cc1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR27 Q9NS67 2/20 0.54
AVPR2 P30518 1/20 0.54
SNCA P37840 1/20 0.48
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
NPC1 O15118 5/20 0.46
RAB9A P51151 4/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 1/20 0.46
KDM4E B2RXH2 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 1/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KLK7 P49862 1/20 0.44
GPR35 Q9HC97 1/20 0.43
PARP1 P09874 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL955495 0.86 LMNA (0.66) NPC1RAB9AHTTSMN1; SMN2LMNA
SCHEMBL5267338 0.84 PPARG (0.48) NPC1RAB9AHTTSMN1; SMN2LMNA
SCHEMBL5265736 0.83 RAB9A (0.49) NPC1RAB9AHTTSMN1; SMN2LMNA
SCHEMBL5266759 0.82 ALDH1A1 (0.46) SNCANPC1RAB9ASMN1; SMN2LMNA
SCHEMBL6544935 0.82 GPR27 (0.72) GPR27AVPR2SNCANPC1RAB9A
SCHEMBL954639 0.81 RAB9A (0.64) NPC1RAB9ALMNATDP1ALDH1A1
SCHEMBL8220374 0.80 KDM4E (0.62) NPC1RAB9AHTTSMN1; SMN2LMNA
SCHEMBL16692879 0.79 LMNA (0.46) SNCANPC1RAB9AHTTLMNA
SCHEMBL954020 0.79 KMT2A (0.52) NPC1RAB9AHTTSMN1; SMN2LMNA
SCHEMBL5265208 0.79 NPC1 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed