SCHEMBL527490

SCHEMBL527490

CCCCCON1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GNAO1 P09471 12/20 0.43
GNAI3 P08754 11/20 0.43
GNAI1 P63096 11/20 0.43
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
SIGMAR1 Q99720 2/20 0.33
LTA4H P09960 1/20 0.32
GBA1 P04062 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374104 0.96 GNAO1 (0.44) GNAO1GNAI3GNAI1HRH2HRH1
SCHEMBL9358034 0.94 GNAO1 (0.40) GNAO1GNAI3GNAI1HRH2HRH1
SCHEMBL27607237 0.88 GNAI3 (0.37) GNAO1GNAI3GNAI1HRH2HRH1
SCHEMBL27507410 0.88 GNAO1 (0.40) GNAO1GNAI3GNAI1
SCHEMBL5312065 0.86 SIGMAR1 (0.37) GNAO1GNAI3GNAI1HRH2HRH1
SCHEMBL27672429 0.85 GNAI3 (0.34) GNAO1GNAI3GNAI1
SCHEMBL4175721 0.82 THRB (0.40) LTA4H
SCHEMBL10378875 0.82 THRB (0.40) LTA4H
SCHEMBL8972630 0.82 THRB (0.40) LTA4H
SCHEMBL4922499 0.82 GNAI3 (0.34) GNAO1GNAI3GNAI1HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150148464-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2015-05-28 US claimed
CN-103025812-B Phosphinic acid hydrazide flame retardant compositions BASF SE 2014-08-13 CN claimed
EP-2598565-B1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2014-04-23 EP claimed
EP-2598565-A1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2013-06-05 EP claimed
US-20130137800-A1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2013-05-30 US claimed
EP-2550321-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2013-01-30 EP claimed
EP-2451869-A1 PHENYLPHOSPHONATE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2012-05-16 EP claimed
US-20120108712-A1 PHENYLPHOSPHONATE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2012-05-03 US claimed
WO-2012013652-A1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2012-02-02 WO claimed
WO-2012013565-A1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2012-02-02 WO claimed
WO-2011117266-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2011-09-29 WO claimed
US-20110237715-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2011-09-29 US claimed
WO-2011003773-A1 PHENYLPHOSPHONATE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2011-01-13 WO claimed
CN-110520413-B Macrocyclic broad spectrum antibiotics 阿奇克斯制药公司 2023-02-17 CN disclosed
US-20150148464-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2015-05-28 US disclosed
CN-103025812-B Phosphinic acid hydrazide flame retardant compositions BASF SE 2014-08-13 CN disclosed
WO-2012013652-A1 PHOSPHINIC ACID HYDRAZIDE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2012-02-02 WO disclosed
WO-2011117266-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2011-09-29 WO disclosed
US-20110237715-A1 FLAME RETARDANT COMPOSITIONS OF PHOSPHINIC ACID SALTS AND NITROXYL DERIVATIVES BASF SE (DE) 2011-09-29 US disclosed
WO-2011003773-A1 PHENYLPHOSPHONATE FLAME RETARDANT COMPOSITIONS BASF SE (DE) 2011-01-13 WO disclosed