SCHEMBL5276249

SCHEMBL5276249

NCCNC(=O)c1cccc(C(=O)CNCCOC(=O)N(c2ccccc2-c2ccccc2)N2CC[CH]CC2)c1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 2/20 0.33
KDM4E B2RXH2 1/20 0.33
KISS1R Q969F8 4/20 0.33
SPHK2 Q9NRA0 1/20 0.33
HTR7 P34969 2/20 0.32
HTR1A P08908 1/20 0.32
CHEK1 O14757 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
F10 P00742 1/20 0.31
TERT O14746 2/20 0.31
LMNA P02545 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272930 0.93 SPHK2 (0.34) KDM4EKISS1RSPHK2ALDH1A1HPGD
SCHEMBL5810881 0.93 SMN1; SMN2 (0.37) SMYD2KDM4EKISS1RSPHK2HTR7
SCHEMBL5277443 0.91 SMN1; SMN2 (0.34) SMYD2KDM4EHTR7HTR1ASMN1; SMN2
SCHEMBL5280997 0.87 CD274 (0.36) ALDH1A1HPGDPDCD1CD274
SCHEMBL5801918 0.87 P2RY12 (0.34) HTR7CHEK1LMNACD274
SCHEMBL5803928 0.86 MAOB (0.35) PDCD1CD274
SCHEMBL5273043 0.86 ALDH1A1 (0.37) ALDH1A1HPGDLMNA
SCHEMBL5281205 0.86 ACKR3 (0.32) CHEK1
SCHEMBL5278178 0.86 ALDH1A1 (0.35) SPHK2ALDH1A1HPGD
SCHEMBL4695511 0.85 PDCD1 (0.34) SMN1; SMN2PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856048-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-11-21 EP claimed
WO-2006098999-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO claimed