SCHEMBL5280997

SCHEMBL5280997

O=C(CNCCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1)c1cccc(C(=O)NCCNCc2ccc(O)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 15/20 0.36
PDCD1 Q15116 11/20 0.36
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
EPHX2 P34913 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5277443 0.90 SMN1; SMN2 (0.34) CD274PDCD1ALDH1A1HPGD
SCHEMBL5276249 0.87 SMYD2 (0.33) CD274PDCD1ALDH1A1HPGD
SCHEMBL5273043 0.87 ALDH1A1 (0.37) ALDH1A1HPGD
SCHEMBL5804676 0.87 ALDH1A1 (0.35) CD274PDCD1ALDH1A1
SCHEMBL6027383 0.87 OPRM1 (0.36) CD274PDCD1ALDH1A1HDAC1
SCHEMBL6027738 0.84 ESRRG (0.40) CD274PDCD1HDAC1
SCHEMBL4692560 0.84 CD274 (0.39) CD274PDCD1HDAC1
SCHEMBL4696335 0.84 PDCD1 (0.44) CD274PDCD1ALDH1A1
SCHEMBL4691952 0.81 PDCD1 (0.35) CD274PDCD1ALDH1A1
SCHEMBL4695511 0.81 PDCD1 (0.34) CD274PDCD1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856048-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-11-21 EP disclosed
WO-2006098999-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO disclosed