SCHEMBL5276265

SCHEMBL5276265

COc1cc2c(cc1OC)CN(CC(=O)N1c3ccccc3Oc3ccccc31)C(C)C2

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.42
P2RX4 Q99571 2/20 0.41
DRD2 P14416 4/20 0.40
DRD4 P21917 4/20 0.40
GFER P55789 1/20 0.40
TSHR P16473 2/20 0.40
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5241484 0.85 BCHE (0.47) MCL1TSHRALDH1A1SMN1; SMN2LMNA
SCHEMBL5242772 0.82 MCL1 (0.44) MCL1P2RX4TSHRALDH1A1SMN1; SMN2
SCHEMBL5243272 0.80 SMN1; SMN2 (0.52) TSHRALDH1A1SMN1; SMN2LMNAHTT
SCHEMBL5242793 0.79 BCHE (0.54) DRD2DRD4ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5278993 0.78 BCHE (0.45) MCL1TSHRALDH1A1LMNAMAPK1
SCHEMBL5279427 0.78 CYP3A4 (0.41) TSHRALDH1A1LMNAHTT
SCHEMBL5288756 0.77 MEN1 (0.54) TSHRALDH1A1KDM4ELMNAHTT
SCHEMBL5276997 0.76 CA2 (0.45) MCL1DRD2CA2CA9ALDH1A1
SCHEMBL5239213 0.74 P2RX4 (0.44) P2RX4KDM4E
SCHEMBL5277209 0.74 CA2 (0.41) MCL1GFERTSHRCA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed