SCHEMBL5276997

SCHEMBL5276997

COc1cc2c(cc1OC)CN(CC(=O)O)C(C)C2

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
RAD52 P43351 1/20 0.43
DRD2 P14416 5/20 0.41
DRD1 P21728 4/20 0.41
ALDH1A1 P00352 2/20 0.41
PDE4B Q07343 1/20 0.41
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
MCL1 Q07820 1/20 0.39
AGTR2 P50052 1/20 0.39
KDM4E B2RXH2 1/20 0.39
DRD5 P21918 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5789193 0.82 CA2 (0.41) CA2CA9DRD2ALDH1A1PDE4B
SCHEMBL5277209 0.81 CA2 (0.41) CA2CA9ALDH1A1KMT2ANPC1
SCHEMBL14376713 0.80 CA2 (0.46) CA2CA9RAD52DRD2DRD1
SCHEMBL5241961 0.78 ADRA2A (0.45) ALDH1A1AGTR2KDM4E
SCHEMBL9425191 0.77 L3MBTL1 (0.51) ALDH1A1KMT2ANPC1KDM4E
SCHEMBL5276265 0.76 MCL1 (0.42) CA2CA9DRD2ALDH1A1MCL1
SCHEMBL5241484 0.76 BCHE (0.47) ALDH1A1KMT2AMCL1
SCHEMBL5242056 0.75 KMT2A (0.45) CA2CA9DRD2ALDH1A1KMT2A
SCHEMBL5786442 0.74 HDAC6 (0.46)
SCHEMBL5289084 0.72 SMN1; SMN2 (0.61) ALDH1A1KMT2ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed