SCHEMBL5280978

SCHEMBL5280978

O=C(CCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1)N(C(=O)NCCNCc1ccc(O)cc1)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 11/20 0.34
PDCD1 Q15116 7/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5271658 0.89 PDCD1 (0.34) CD274PDCD1
SCHEMBL5271781 0.87 PTGIR (0.31)
SCHEMBL6021284 0.85 LTB4R2 (0.37) CD274PDCD1
SCHEMBL5805321 0.83 HDAC3 (0.40)
SCHEMBL6021999 0.82 LTB4R2 (0.33) CD274PDCD1
SCHEMBL6022022 0.82 CHRM2 (0.39) CD274PDCD1
SCHEMBL6027475 0.80 TRPV1 (0.37)
SCHEMBL6021982 0.80 ALDH1A1 (0.39)
SCHEMBL6021934 0.80 MEN1 (0.40)
SCHEMBL6022017 0.79 HTR1A (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006098997-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO claimed
EP-1856048-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-11-21 EP disclosed
WO-2006098999-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO disclosed
WO-2006098997-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO disclosed
WO-2006099091-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO disclosed