SCHEMBL6021999

SCHEMBL6021999

O=C(CCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1)N(CNCc1ccc(O)cc1)Cc1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 4/20 0.33
ALDH1A1 P00352 3/20 0.32
SLC6A4 P31645 2/20 0.32
CCR6 P51684 1/20 0.31
PAX8 Q06710 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
HTR5A P47898 2/20 0.31
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30
DRD4 P21917 2/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
ADRA1B P35368 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6021284 0.89 LTB4R2 (0.37) LTB4R2ALDH1A1PDCD1CD274LMNA
SCHEMBL6021982 0.83 ALDH1A1 (0.39) ALDH1A1TRPV1LMNA
SCHEMBL6022017 0.83 HTR1A (0.36) ALDH1A1TRPV1HTR5AHTR1ADRD2
SCHEMBL6022022 0.82 CHRM2 (0.39) ALDH1A1CCR6PAX8HTR1ADRD2
SCHEMBL5280978 0.82 CD274 (0.34) PDCD1CD274
SCHEMBL6027475 0.80 TRPV1 (0.37) TRPV1HTR1ADRD2HTR7HTR6
SCHEMBL6021934 0.80 MEN1 (0.40) ALDH1A1TRPV1
SCHEMBL6022221 0.79 BCHE (0.39) TRPV1HTR5AHTR1ADRD2HTR7
SCHEMBL6028157 0.79 ACHE (0.39) LTB4R2ALDH1A1CCR6PAX8HTR1A
SCHEMBL6027362 0.77 TRPV1 (0.39) ALDH1A1TRPV1PDCD1CD274SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723110-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP claimed
WO-2005087735-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO claimed
EP-1723110-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP disclosed
WO-2005087735-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO disclosed