SCHEMBL6027475

SCHEMBL6027475

O=C(CCc1ccc(CNCc2ccc(O)cc2)cc1)NCCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.37
CNR2 P34972 1/20 0.35
GAA P10253 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
HPGD P15428 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
SLC6A5 Q9Y345 1/20 0.34
HTR7 P34969 4/20 0.34
HTR1A P08908 3/20 0.34
DRD2 P14416 3/20 0.34
HTR6 P50406 3/20 0.34
HCAR2 Q8TDS4 2/20 0.33
LTA4H P09960 1/20 0.33
EPHX2 P34913 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695551 0.93 CNR2 (0.40) TRPV1CNR2GAAKDM4ELMNA
SCHEMBL4691773 0.90 KDM4E (0.41) CNR2KDM4ELMNAHPGDHTR7
SCHEMBL4695176 0.90 POLB (0.37) CNR2KDM4ELMNAHPGDLTA4H
SCHEMBL4692631 0.90 ALDH1A1 (0.35) TRPV1CNR2KDM4ELMNAERCC1
SCHEMBL6027362 0.90 TRPV1 (0.39) TRPV1LMNAOPRM1OPRD1OPRK1
SCHEMBL5805321 0.88 HDAC3 (0.40) TRPV1SLC6A5HTR7HTR1ADRD2
SCHEMBL6022221 0.85 BCHE (0.39) TRPV1ERCC1ERCC4HTR7HTR1A
SCHEMBL6021982 0.85 ALDH1A1 (0.39) TRPV1GAALMNALTA4HEPHX2
SCHEMBL6021934 0.85 MEN1 (0.40) TRPV1GAALTA4HEPHX2
SCHEMBL6022017 0.84 HTR1A (0.36) TRPV1GAAHTR7HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723108-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP claimed
WO-2005087733-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO claimed