SCHEMBL4691952

SCHEMBL4691952

NC(=O)CNCc1ccc(C(=O)CNCCOC(=O)N(c2ccccc2-c2ccccc2)N2CC[CH]CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 4/20 0.35
CD274 Q9NZQ7 4/20 0.35
ALDH1A1 P00352 2/20 0.34
SPHK2 Q9NRA0 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
LMNA P02545 1/20 0.34
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
SCN3A Q9NY46 1/20 0.32
S1PR1 P21453 5/20 0.31
LTA4H P09960 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696335 0.92 PDCD1 (0.44) PDCD1CD274ALDH1A1LTA4H
SCHEMBL4692560 0.90 CD274 (0.39) PDCD1CD274S1PR1LTA4H
SCHEMBL4695511 0.90 PDCD1 (0.34) PDCD1CD274DPP4
SCHEMBL4697200 0.89 HDAC1 (0.37) PDCD1CD274ALDH1A1LMNA
SCHEMBL6027383 0.88 OPRM1 (0.36) PDCD1CD274ALDH1A1LMNAOPRM1
SCHEMBL4694658 0.87 ALDH1A1 (0.36) PDCD1CD274ALDH1A1SPHK2SPHK1
SCHEMBL4696628 0.86 HDAC1 (0.35) PDCD1CD274LTA4H
SCHEMBL12505524 0.85 ALDH1A1 (0.34) ALDH1A1
SCHEMBL4692631 0.85 ALDH1A1 (0.35) ALDH1A1SPHK2SPHK1LMNAOPRM1
SCHEMBL4694768 0.85 HDAC1 (0.36) LMNALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP claimed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO claimed