SCHEMBL5282008

SCHEMBL5282008

O=C(O)Nc1ccc(SCC(=O)NCCc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.56
MEN1 O00255 5/20 0.56
KMT2A Q03164 5/20 0.56
CNR1 P21554 1/20 0.55
ALDH1A1 P00352 6/20 0.53
HTT P42858 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
LMNA P02545 2/20 0.53
MAOA P21397 1/20 0.53
MAOB P27338 1/20 0.53
CYP3A4 P08684 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C9 P11712 2/20 0.51
TP53 P04637 1/20 0.51
MAPK1 P28482 1/20 0.51
HSP90AA1 P07900 1/20 0.51
XBP1 P17861 1/20 0.51
ALOX12 P18054 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CA12 O43570 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6037988 0.84 MMP1 (0.51) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL5277895 0.76 CYP2C9 (0.58) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL1695076 0.76 SMN1; SMN2 (0.66) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL6038318 0.76 HDAC3 (0.58) MAPTMEN1KMT2AALDH1A1HTT
SCHEMBL20303790 0.75 MAPT (0.61) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL152811 0.74 KMT2A (0.74) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL15306496 0.73 CNR1 (0.77) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL15306499 0.73 CNR1 (0.77) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL1395699 0.73 CNR1 (0.60) MAPTMEN1KMT2ACNR1ALDH1A1
SCHEMBL20718868 0.73 ALDH1A1 (0.60) MAPTMEN1KMT2ACNR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863804-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2007-12-12 EP disclosed
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO disclosed