SCHEMBL5282202

SCHEMBL5282202

CCCCCN(NCc1ccc2c(c1)CCO2)C(=O)CCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 8/20 0.38
CHRM1 P11229 8/20 0.38
CHRM4 P08173 3/20 0.38
CHRM3 P20309 3/20 0.38
CHRM2 P08172 2/20 0.37
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
GSK3B P49841 1/20 0.35
FAAH O00519 1/20 0.33
SLC6A9 P48067 1/20 0.33
EDNRB P24530 1/20 0.32
ATM Q13315 1/20 0.32
RYR2 Q92736 1/20 0.31
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CXCR3 P49682 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5283848 0.90 DAGLA (0.35) KDM1AMAOAMAOB
SCHEMBL6021930 0.80 LTB4R2 (0.34)
SCHEMBL6022345 0.78 CYP1A2 (0.37)
SCHEMBL5285440 0.74 CHRM3 (0.58) CHRM3
SCHEMBL5276883 0.69 CHRM3 (0.33) CHRM3RAB9ANPC1
SCHEMBL6022322 0.68 ADRB2 (0.35) CHRM1CHRM3CHRM2
SCHEMBL4691377 0.67 KMT2A (0.36) RAB9ANPC1
SCHEMBL6021999 0.67 LTB4R2 (0.33)
SCHEMBL5801465 0.66 MEN1 (0.34) CHRM3RAB9APOLB
SCHEMBL5803533 0.66 ERCC1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866284-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-12-19 EP disclosed
WO-2006099167-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO disclosed