SCHEMBL6022322

SCHEMBL6022322

CN(CCCCCNCCc1ccc(O)cc1)C(=O)CCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.35
CHRM3 P20309 3/20 0.35
CHRM2 P08172 5/20 0.35
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OPRK1 P41145 2/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
DRD1 P21728 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
PTGS2 P35354 1/20 0.32
HRH1 P35367 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6022022 0.93 CHRM2 (0.39) ADRB2CHRM3CHRM2BCHEACHE
SCHEMBL6028157 0.87 ACHE (0.39) ADRB2CHRM3CHRM2BCHEACHE
SCHEMBL5247685 0.85 OPRK1 (0.37) ADRB2OPRK1ADORA3CHRM1ADRA2B
SCHEMBL6023018 0.84 SLC6A5 (0.38) KDM4ESMN1; SMN2OPRK1OPRM1OPRD1
SCHEMBL6021930 0.84 LTB4R2 (0.34) OPRM1
SCHEMBL5805321 0.81 HDAC3 (0.40) BCHE
SCHEMBL6022468 0.80 ADRB2 (0.43) ADRB2KDM4ESMN1; SMN2OPRK1ADORA3
SCHEMBL6021287 0.80 HTR1A (0.36)
SCHEMBL5281472 0.80 TAAR1 (0.37) CHRM3KDM4EALDH1A1SMN1; SMN2CHRM1
SCHEMBL6021934 0.79 MEN1 (0.40) ADRB2CHRM3BCHEALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723111-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-11-22 EP disclosed
WO-2005087732-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2005-09-22 WO disclosed