SCHEMBL528413

SCHEMBL528413

CCCC(C(=O)NC)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
KCNQ2 O43526 2/20 0.53
ALDH1A1 P00352 2/20 0.50
CRHBP P24387 2/20 0.49
CRHR2 Q13324 2/20 0.49
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
POLB P06746 2/20 0.46
GPR88 Q9GZN0 1/20 0.46
HDAC3 O15379 3/20 0.46
HDAC4 P56524 3/20 0.46
HDAC1 Q13547 3/20 0.46
HDAC7 Q8WUI4 3/20 0.46
HDAC2 Q92769 3/20 0.46
HDAC10 Q969S8 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2049579 0.85 ALDH1A1 (0.66) CYP1A2CYP3A4CYP2C9KCNQ2ALDH1A1
SCHEMBL8113733 0.84 CTSD (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7504901 0.84 LMNA (0.49) KCNQ2ALDH1A1CRHBPCRHR2LMNA
SCHEMBL2721958 0.81 LMNA (0.50) KCNQ2ALDH1A1CRHBPCRHR2LMNA
SCHEMBL10573413 0.81 HTR2A (0.53) CYP3A4CYP2C19ALDH1A1LMNA
SCHEMBL19228532 0.81 CYP2C19 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL643461 0.81 CYP2C19 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14423896 0.80 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9055208 0.80 ROCK2 (0.50) ALDH1A1CRHBPCRHR2LMNAHTT
SCHEMBL19256857 0.80 ROCK2 (0.50) ALDH1A1CRHBPCRHR2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006433-B2 Substituted pyrimidines MERCK SHARP & DOHME CORP. (US) 2015-04-14 US disclosed