SCHEMBL5286006

SCHEMBL5286006

N#Cc1ccccc1S(=O)(=O)c1ccc(CO)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.57
ABCC9 O60706 3/20 0.50
ABCC8 Q09428 3/20 0.50
KCNJ11 Q14654 3/20 0.50
KCNJ8 Q15842 3/20 0.50
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.45
HTT P42858 1/20 0.45
LMNA P02545 2/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5284219 0.84 HSD11B1 (0.53) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3163460 0.84 HSD11B1 (0.47) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL1146161 0.81 HSD11B1 (0.59) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL28539914 0.79 HSD11B1 (0.61) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL4159366 0.79 HSD11B1 (0.57) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3157029 0.79 HSD11B1 (0.57) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL28541788 0.79 HSD11B1 (0.61) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3263174 0.78 POLB (0.52) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8514629 0.77 ALDH1A1 (0.62) HSD11B1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL30468568 0.77 ALDH1A1 (0.62) HSD11B1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861079-A1 ARYLSULFONYL BENZYL ETHERS AS 5-HT2A ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 2007-12-05 EP disclosed
WO-2006097766-A1 ARYLSULFONYL BENZYL ETHERS AS 5-HT2A ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 2006-09-21 WO disclosed