SCHEMBL5286958

SCHEMBL5286958

O=C(O)NCCC(O)c1cccs1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
KMT2A Q03164 1/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KEAP1 Q14145 1/20 0.42
HTR1A P08908 1/20 0.39
KDM4E B2RXH2 1/20 0.39
TP53 P04637 3/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
CYP2C19 P33261 1/20 0.38
SLC5A2 P31639 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15064090 0.83 NPC1 (0.51) RAB9ANPC1KMT2ACES2CES1
SCHEMBL12546521 0.83 L3MBTL1 (0.41) RAB9ANPC1KMT2ACES2CES1
SCHEMBL1946731 0.83 L3MBTL1 (0.41) RAB9ANPC1KMT2ACES2CES1
SCHEMBL13649162 0.80 LMNA (0.53) KEAP1LMNASMN1; SMN2POLB
SCHEMBL13655772 0.80 LMNA (0.53) KEAP1LMNASMN1; SMN2POLB
SCHEMBL4440609 0.78 NPC1 (0.57) RAB9ANPC1KMT2ACES2CES1
SCHEMBL165478 0.78 SLC6A2 (0.49) RAB9ANPC1KMT2AHTR1ACYP2C19
SCHEMBL98019 0.78 SLC6A2 (0.49) RAB9ANPC1KMT2AHTR1ACYP2C19
SCHEMBL1201347 0.78 SLC6A2 (0.49) RAB9ANPC1KMT2AHTR1ACYP2C19
SCHEMBL6499256 0.78 NPC1 (0.48) RAB9ANPC1KMT2ACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070116643-A1 Novel aryloxypropanamines CONCERT PHARMACEUTICALS INC. (US) 2007-05-24 US disclosed
WO-2007005644-A2 NOVEL ARYLOXYPROPANAMINES CONCERT PHARMACEUTICALS INC. (US) 2007-01-11 WO disclosed