SCHEMBL5287728

SCHEMBL5287728

CCOC(=O)CNc1cccc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.54
GAA P10253 2/20 0.54
TRPV1 Q8NER1 1/20 0.54
ALDH1A1 P00352 8/20 0.50
LMNA P02545 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
EGFR P00533 1/20 0.50
TSHR P16473 1/20 0.50
KDM4E B2RXH2 5/20 0.49
HTT P42858 3/20 0.49
THRB P10828 1/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
MAPK1 P28482 1/20 0.48
RAB9A P51151 1/20 0.48
HPGD P15428 1/20 0.48
KYAT1 Q16773 1/20 0.48
EPHX2 P34913 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11355645 0.89 POLB (0.55) MAPTGAAALDH1A1LMNASMN1; SMN2
SCHEMBL7593370 0.86 MEN1 (0.51) MAPTGAAALDH1A1LMNASMN1; SMN2
SCHEMBL1120688 0.85 MAPT (0.59) MAPTGAATRPV1ALDH1A1LMNA
SCHEMBL1751588 0.85 MAPT (0.56) MAPTGAATRPV1ALDH1A1LMNA
SCHEMBL29860111 0.84 MAPT (0.53) MAPTGAAALDH1A1LMNAHTT
SCHEMBL8168563 0.84 MAPT (0.53) MAPTGAAALDH1A1LMNAHTT
Hydrochloric Acid SCHEMBL15646288 0.84 MEN1 (0.50) MAPTGAAALDH1A1LMNASMN1; SMN2
SCHEMBL9271365 0.84 HTT (0.50) MAPTGAATRPV1ALDH1A1LMNA
SCHEMBL6239200 0.84 KMT2A (0.47) MAPTGAAALDH1A1LMNAKDM4E
SCHEMBL11729327 0.84 MEN1 (0.51) MAPTGAAALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250049804-A1 FERROCHELATASE INHIBITORS AND METHODS OF USE UNIV INDIANA RES & TECH CORP (US) 2025-02-13 US disclosed
US-12161642-B2 Ferrochelatase inhibitors and methods of use INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2024-12-10 US disclosed
CN-110372627-B 1,3, 4-oxadiazole derivative and preparation method and application thereof 南昌大学 2022-12-06 CN disclosed
US-20210121465-A1 FERROCHELATASE INHIBITORS AND METHODS OF USE GACHON UNIVERSITY OF INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2021-04-29 US disclosed
US-20070135499-A1 Hydrazide compounds AERIE PHARMACEUTICALS, INC. (US) 2007-06-14 US disclosed
US-20070135499-A1 Hydrazide compounds AERIE PHARMACEUTICALS, INC. (US) 2007-06-14 US disclosed
US-20070135499-A1 Hydrazide compounds AERIE PHARMACEUTICALS, INC. (US) 2007-06-14 US disclosed
WO-2007008942-A2 PHENYLAMINO-ACETIC ACID [1-(PYRIDIN-4-YL)-METHYLIDENE]-HYDRAZIDE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS OF G PROTEIN-COUPLED RECEPTOR KINASES FOR THE TREATMENT OF EYE DISEASES AERIE PHARMACEUTICALS, INC. (US) 2007-01-18 WO disclosed
US-4237132-A ARTERIOSCLEROSIS, ANTICHOLESTEROL, ANTILIPEMIC NIPPON SHINYAKU CO., LTD. (JP) 1980-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250049804-A1 FERROCHELATASE INHIBITORS AND METHODS OF USE FECH, SLC40A1, TPI1 MAPT 3197/4885GAA 170/4885TRPV1 2992/4885
US-20070135499-A1 Hydrazide compounds GRK4, GRK2, GRK1 MAPT 3473/4885GAA 997/4885TRPV1 108/4885
US-20210121465-A1 FERROCHELATASE INHIBITORS AND METHODS OF USE FECH, SLC40A1, TPI1 MAPT 3197/4885GAA 170/4885TRPV1 2992/4885
US-12161642-B2 Ferrochelatase inhibitors and methods of use FECH, SLC40A1, TPI1 MAPT 3197/4885GAA 170/4885TRPV1 2992/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.