SCHEMBL5290607

SCHEMBL5290607

COc1nsc(S(=O)(=O)Cc2ccccc2C)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
GAA P10253 1/20 0.49
LMNA P02545 4/20 0.45
GRM4 Q14833 1/20 0.38
NPC1 O15118 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
RAB9A P51151 1/20 0.34
TLR9 Q9NR96 2/20 0.34
TXNRD1 Q16881 1/20 0.33
HSP90AA1 P07900 1/20 0.33
CXCR5 P32302 1/20 0.33
APLNR P35414 1/20 0.33
CCR6 P51684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5301629 0.75 KMT2A (0.41) ALDH1A1GRM4NPSR1CYP3A4CYP2D6
SCHEMBL5290581 0.75 PLCG1 (0.47) ALDH1A1LMNAGRM4NPSR1CYP3A4
SCHEMBL5295830 0.75 L3MBTL1 (0.32) TXNRD1
SCHEMBL5298171 0.74 TXNRD1 (0.45) ALDH1A1LMNAGRM4NPSR1CYP1A2
SCHEMBL5303247 0.74 CYP2A6 (0.37) HTT
SCHEMBL5306337 0.73 TXNRD1 (0.49) ALDH1A1LMNAGRM4TXNRD1TP53
SCHEMBL5295817 0.73 CDC25A (0.45) ALDH1A1GAALMNANPC1MEN1
SCHEMBL5297846 0.73 AR (0.45) LMNANPC1MEN1KMT2ARAB9A
SCHEMBL5290295 0.70 MRGPRX4 (0.43) MEN1KMT2ARAB9ATP53HTT
SCHEMBL5293863 0.70 AKR1B1 (0.46) GAALMNAGRM4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO claimed
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed