SCHEMBL5303247

SCHEMBL5303247

COc1nsc(S(=O)(=O)Cc2nccc3ccccc23)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
PLAU P00749 3/20 0.33
PLG P00747 1/20 0.33
MMP1 P03956 1/20 0.32
MMP13 P45452 1/20 0.32
ADAM17 P78536 1/20 0.32
F12 P00748 1/20 0.31
NCF1 P14598 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
BACE1 P56817 1/20 0.31
EGFR P00533 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SCN9A Q15858 1/20 0.30
CASP3 P42574 1/20 0.30
SENP6 Q9GZR1 1/20 0.30
TUBB4A P04350 1/20 0.30
TUBB P07437 1/20 0.30
TUBA3C P0DPH7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5363871 0.83 PLAU (0.41) CYP2A6PLAUPLGF12NCF1
SCHEMBL5293941 0.77 TXNRD1 (0.43) HTT
SCHEMBL28239901 0.74 CYP2A6 (0.47) CYP2A6PLAUPLGMMP1MMP13
SCHEMBL5290607 0.74 ALDH1A1 (0.49) HTT
SCHEMBL5369139 0.71 L3MBTL1 (0.47) MMP13SMN1; SMN2HTT
SCHEMBL5301629 0.71 KMT2A (0.41) MMP1ADAM17SMN1; SMN2
SCHEMBL5297846 0.71 AR (0.45) SMN1; SMN2
SCHEMBL5295830 0.70 L3MBTL1 (0.32)
SCHEMBL5290581 0.70 PLCG1 (0.47) MMP1MMP13SMN1; SMN2HTT
SCHEMBL5288284 0.70 TXNRD1 (0.47) SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO claimed
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed