SCHEMBL5301071

SCHEMBL5301071

O=S(=O)(Cc1ccc2c(c1)OCO2)c1ncns1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.42
CYP2D6 P10635 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A1 P30531 1/20 0.42
SLC6A3 Q01959 1/20 0.42
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
CMA1 P23946 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
CYP1A2 P05177 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
CYP2C19 P33261 1/20 0.40
GFER P55789 1/20 0.39
SLC6A4 P31645 1/20 0.39
MAPT P10636 1/20 0.39
PDE5A O76074 2/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306349 0.77 ALDH1A1 (0.43) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3
SCHEMBL5293205 0.76 TAAR1 (0.43) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3
SCHEMBL5293214 0.74 HSD17B10 (0.40) CYP2D6SLC6A2SLC6A3ALDH1A1GAA
SCHEMBL5294272 0.73 POLB (0.46) CYP3A4CYP2D6ALDH1A1CYP2C19MAPT
SCHEMBL30311564 0.70 TAAR1 (0.56) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3
SCHEMBL924831 0.70 ALDH1A1 (0.54) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3
SCHEMBL5286204 0.70 KCNH2 (0.44) ALDH1A1GAAHSD17B10L3MBTL1LMNA
SCHEMBL5308656 0.70 MEN1 (0.42) CYP3A4CYP2D6SLC6A2ALDH1A1GAA
SCHEMBL6529898 0.70 TAAR1 (0.55) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3
SCHEMBL6528293 0.69 ALDH1A1 (0.52) CYP3A4CYP2D6SLC6A2SLC6A1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO claimed
WO-2007012724-A1 1,2,4-THIADIAZOLE DERIVATIVES ANTIFUNGAL COMPOUNDS, COMPOSITIONS CONTAINING SAID COMPOUNDS AND THE USE THEREOF CYTOMICS SYSTEMS (FR) 2007-02-01 WO disclosed