SCHEMBL5306266

SCHEMBL5306266

NCC1CCN(CCCS(=O)(=O)N2CCNCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 14/20 0.47
GNAO1 P09471 4/20 0.38
GNAI3 P08754 3/20 0.36
GNAI1 P63096 3/20 0.36
NCF1 P14598 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212310 0.84 NCF1 (0.49) HTR4GNAO1GNAI3GNAI1NCF1
SCHEMBL5215771 0.83 HTR4 (0.47) HTR4NCF1
SCHEMBL5216687 0.82 HTR4 (0.48) HTR4GNAO1GNAI3GNAI1NCF1
SCHEMBL5214688 0.82 HTR4 (0.48) HTR4NCF1
SCHEMBL5215967 0.82 HTR4 (0.48) HTR4NCF1
SCHEMBL5219363 0.81 HTR4 (0.48) HTR4GNAO1GNAI3GNAI1NCF1
SCHEMBL5306262 0.81 HTR4 (0.46) HTR4GNAO1GNAI3GNAI1
SCHEMBL5218999 0.80 HTR4 (0.49) HTR4NCF1
SCHEMBL5214555 0.78 HTR4 (0.41) HTR4NCF1
SCHEMBL960926 0.76 HTR4 (0.43) HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112270-B1 DIHYDROBENZODIOXINE CARBOXAMIDE AND KETONE DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed