SCHEMBL5313176

SCHEMBL5313176

COc1cccc(Cn2nc(C)c(-c3ccccc3OCc3ccccc3)c(CCc3ccccc3)c2=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.47
HTR1A P08908 2/20 0.47
DRD2 P14416 2/20 0.47
ALDH1A1 P00352 2/20 0.46
FAAH O00519 1/20 0.46
MGLL Q99685 1/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
CYP1A2 P05177 4/20 0.45
CYP3A4 P08684 4/20 0.45
CYP2C19 P33261 4/20 0.45
CYP2C9 P11712 3/20 0.45
TSHR P16473 3/20 0.45
CYP2D6 P10635 2/20 0.45
PDE5A O76074 1/20 0.45
FPR2 P25090 1/20 0.42
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5308221 0.88 ALDH1A1 (0.42) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5313082 0.86 LMNA (0.45) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5311498 0.86 ALDH1A1 (0.51) ALDH1A1FAAHGAAPKMCYP1A2
SCHEMBL5308884 0.83 ALDH1A1 (0.44) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5308888 0.83 ALDH1A1 (0.44) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5308868 0.79 GAA (0.42) ALDH1A1GAAPKMCYP1A2CYP3A4
SCHEMBL5311126 0.79 ALDH1A1 (0.42) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5311122 0.79 ALDH1A1 (0.42) ABCB1HTR1ADRD2ALDH1A1FAAH
SCHEMBL5307948 0.79 CASR (0.49) ALDH1A1GAAPKMPDE5AFPR2
SCHEMBL5307935 0.79 TP53 (0.44) ALDH1A1MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed