SCHEMBL5308221

SCHEMBL5308221

COc1cc(Cn2nc(C)c(-c3ccccc3OCc3ccccc3)c(CCc3cccc(F)c3)c2=O)cc(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ABCB1 P08183 6/20 0.41
HTR1A P08908 2/20 0.41
DRD2 P14416 2/20 0.41
CASR P41180 2/20 0.39
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
MAPK14 Q16539 2/20 0.38
MAOB P27338 2/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5313082 0.93 LMNA (0.45) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5313176 0.88 ABCB1 (0.47) ALDH1A1HTTSMN1; SMN2ABCB1HTR1A
SCHEMBL5307935 0.87 TP53 (0.44) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5315681 0.86 CASR (0.49) ALDH1A1HTTCASRGAAPKM
SCHEMBL5316086 0.84 CASR (0.41) ALDH1A1HTTCASRGRIN1GRIN2B
SCHEMBL5311481 0.83 ALDH1A1 (0.40) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5311478 0.83 ALDH1A1 (0.40) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5312354 0.83 TP53 (0.42) ALDH1A1MEN1LMNAHTTKMT2A
SCHEMBL5308342 0.83 POLB (0.48) ALDH1A1MEN1LMNAKMT2ASMN1; SMN2
SCHEMBL5310887 0.82 LMNA (0.38) ALDH1A1MEN1LMNAHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed